Showing posts with label Inverse Agonists. Show all posts
Showing posts with label Inverse Agonists. Show all posts

Sunday, May 9, 2021

Inverse Agonists

Inverse agonists are drugs that have affinity at the receptor site but produce opposite actions (turn “off” a receptor that is activated or turn “on” a receptor that is not currently active). When two or more agonists are administered together, a competition for drug-receptor binding sites occurs.